Papers - Sugai, Takeshi

Structure–activity relationship of celecoxib and rofecoxib for the membrane permeabilizing activity

N. Yamakawa, K. Suzuki, Y. Yamashita, T. Katsu, K. Hanaya, M. Shoji, T. Sugai and T. Mizushima

Bioorg. Med. Chem. 22   2529–2534 2014.04

Research paper (scientific journal), Joint Work, Accepted

Divergent synthesis of pseudoenantiomers for ABC-ring moiety of steroids

M. Furuta, K. Hanaya, T. Sugai and M. Shoji

Tetrahedron Lett. 55   3189–3191 2014.02

Research paper (scientific journal), Joint Work, Accepted

Stereoselective Synthesis of Scyphostatin Hydrophilic Moiety

K. Kuwata, M. Suzuki, Y. Inami, K. Hanaya, T. Sugai and M. Shoji

Tetrahedron Lett. 55   2856–2858 2014.02

Research paper (scientific journal), Joint Work, Accepted

(-)-Benzyl 2,3-dideoxy-β-D-erythro-hex-2-enopyranoside

S. Ohba, H. Okazaki, Y. Ueda, K. Hanaya and T. Sugai

Acta Cryst. E69   o1811 2013.12

Research paper (scientific journal), Joint Work, Accepted

Whole-cell yeast-mediated preparation of (R)-2-chloro-1-(3-nitrophenyl)ethanol as a synthetic precursor for (R)-phenylephrine

D. Tokoshima, K. Hanaya, M. Shoji and T. Sugai

J. Mol. Catal. B: Enz. 97   95-99 2013.12

Research paper (scientific journal), Joint Work, Accepted

Synthesis of (R)-bambuterol based on asymmetric reduction of 1-[3,5-bis(dimethylcarbamoyloxy)phenyl]-2-chloroethanone with incubated whole cells of Williopsis californica JCM 3600

K. Asami, T. Machida, S. Jung, K. Hanaya, M. Shoji and T. Sugai

J. Mol. Catal. B: Enz. 97   106-109 2013.12

Research paper (scientific journal), Joint Work, Accepted

Synthesis of Methyl epi-Anhydroquinate Utilizing [2,3]-Sigmatropic Rearrangement of Iodosoalkene

S. Inomata, M. Ueda, T. Sugai and M. Shoji

Chem. Lett. 42   1273-1275 2013.10

Research paper (scientific journal), Joint Work, Accepted

An expeditious route for 2-acetamido-4-O-methyl-2-deoxy-D-mannopyranose from a Ferrier derivative of tri-O-acetyl-D-glucal, which contributes to the synthesis of laninamivir (CS-8958), a neuraminidase inhibitor

H. Okazaki, K. Hanaya, M. Shoji and T. Sugai

Tetrahedron 69   7931-7935 2013.09

Research paper (scientific journal), Joint Work, Accepted

Chemo-enzymatic enantioconvergent approach toward ethyl shikimate from ethyl 5-hydroxy-3,4-isopropylidenedioxycyclohex-1-enecarboxylate

Y. Yamashita, K. Hanaya, T. Sugai, T. Mizushima and M. Shoji

Tetrahedron 69   6527-6532 2013.08

Research paper (scientific journal), Joint Work, Accepted

Formal synthesis of (+)-madindoline A, a potent IL-6 inhibitor, utilizing enzymatic discrimination of quaternary carbon

K. Shimizu, M. Tomita, K. Fuhshuku, T. Sugai and M. Shoji

Nat. Prod. Commun. 8   897-901 2013.07

Research paper (scientific journal), Joint Work, Accepted

Synthesis of okicamelliaside, a glucoside of ellagic acid with potent anti-degranulation activity

R. Kobayashi, K. Hanaya, M. Shoji, S. Ohba and T. Sugai

Biosci. Biotechnol. Biochem. 77   810-813 2013.06

Research paper (scientific journal), Joint Work, Accepted

Chemo-enzymatic transformation of naturally abundant naringin to luteolin, a flavonoid with various biological effects

R. Kobayashi, T. Itou, K. Hanaya, M. Shoji, N. Hada and T. Sugai

J. Mol. Catal. B: Enz. 92   14-18 2013.06

Research paper (scientific journal), Joint Work, Accepted

Stereoselective construction of cis-decalin framework via radical domino cyclization

E. Suzuki, M. Ueda, S. Ohba, T. Sugai　and M. Shoji

Tetrahedron Lett. 54   1589-1592 2013.02

Research paper (scientific journal), Joint Work, Accepted

Triazoyl–phenyl linker system enhancing the aqueous solubility of a molecular probe and its efficiency in affinity labeling of a target protein for jasmonate glucoside

S. Tamura, S. Inomata, M. Ebine, T. Genji, I. Iwakura, M. Mukai, M. Shoji, T. Sugai and M. Ueda

Bioorg. Med. Chem. Lett. 23   188-193 2013.01

Research paper (scientific journal), Joint Work, Accepted

A Chemo-enzymatic Expeditious Route to Racemic Dihexanoyl (2R*,3R*,4R*)-DHMEQ (Dehydroxymethylepoxyquinomycin), the Precursor for Lipase-catalyzed Synthesis of (2S,3S,4S)-DHMEQ, a Potent NF-kB Inhibitor

R. Kobayashi, K. Hanaya, M. Shoji, K. Umezawa　and T. Sugai

Chem. Pharm. Bull. 60   1220-1223 2012.12

Research paper (scientific journal), Joint Work, Accepted

Chemo-enzymatic routes for (R)-terbutaline hydrochloride based on microbial asymmetric reduction of a-haloacetophenones

S. Taketomi, M. Asano, T. Higashi, M. Shoji　and T. Sugai

J. Mol. Catal. B: Enz. 84   83-88 2012.10

Research paper (scientific journal), Joint Work, Accepted

Reduction of acetophenones with methyl fluorines and a bulky group on the aromatic ring using microorganisms and related enzymes

C. Abe, T. Sugawara, T. Machida, T. Higashi, K. Hanaya, M. Shoji, C. Cao, T. Yamamoto, T. Matsuda and T. Sugai

J. Mol. Catal. B: Enz. 82   86-91 2012.08

Research paper (scientific journal), Joint Work, Accepted

Stereoselective approach to (2R,3S)- and (2R,3R)-1,2-(cyclohexylidenedioxy)hept-6-en-3-ol by microbial reduction

M. Furuta, M. Shoji　and T. Sugai

J. Mol. Catal. B: Enz. 82   8-11 2012.07

Research paper (scientific journal), Joint Work, Accepted

A Phthalimide derivative that Inhibits centrosomal clustering is effective on multiple myeloma

H. Shiheido, F. Terada, N. Tabata, I. Hayakawa, N. Matsumura, H. Takashima, Y. Ogawa, W, Du, T. Yamada, M. Shoji, T. Sugai, N. Doi, S. Ijima, Y. Hattori　and H. Yanagawa

Plos One 7   e38878 2012.06

Research paper (scientific journal), Joint Work, Accepted

Hybrid stereoisomers of a compact molecular probe based on a jasmonic acid glucoside: Syntheses, and biological evaluations

M. Ueda, G. Q. Yang, Y. Ishimaru, T. Itabashi, S. Tamura, H. Kiyota, S. Kuwahara, S. Inomata, M. Shoji and T. Sugai

Bioorg. Med. Chem. 20   5832-5843 2012.04

Research paper (scientific journal), Joint Work, Accepted