Papers - Takahashi, Daisuke

Total Synthesis of Mono-Rhamnolipids Using Organophotoacid-Catalyzed Glycosylation and Their Antibacterial Activity

Kohei Higashiyama, Kanae Hosomi, Kazuki Senoo, Chigusa Hayashi, Masayuki Igarashi, *DAISUKE TAKAHASHI, *K. Toshima

CHEMICAL COMMUNICATIONS (Royal Society of Chemistry)   2025.12

Research paper (scientific journal), Joint Work, Corresponding author, Accepted

Synthesis and structure-activity relationship of azithromycin derivatives against non-tuberculous mycobacteria

Yuka Isozaki, Ali Ahsan Muzahid, Tatsuki Wakata, Maho Fujino, Yoshikazu Tanaka, Chigusa Hayashi, Yoshimasa Ishizaki, Tomokazu Ohishi, Ayumi Morita, Shunichi Ohba, Takeshi Yokoyama, *Masayuki Igarashi, *Kazunobu Toshima, *DAISUKE TAKAHASHI

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Elsevier)  304   118520 2025.12

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted

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Glycosylation Using Diethyl Phosphite Donor Activated by Edible Polyphenol Ellagic Acid

Hidenari Shigeta, Ayato Watanabe, Chikako Shiraishi, DAISUKE TAKAHASHI, *Kazunobu Toshima

CARBOHYDRATE RESEARCH (Elsevier)  558   109712 (6 pages) 2025.10

Research paper (scientific journal), Joint Work, Accepted

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Inhibitory Effect of Fucoidan Analogs on Highly Metastatic Gastric Cancer Cells via Galectin-4 Inhibition

Shuting Ji, Maniyamma Aswathy, Yuya Kuboki, Yoshio Takada, Kazunobu Toshima, DAISUKE TAKAHASHI, *Hiroko Ideo

INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (MDPI)  26 ( 18 ) 9228 - 9228 2025.09

Research paper (scientific journal), Joint Work, Accepted

An alkaline phosphatase-activatable photosensitizer based on 2-anthrol for selective targeting of cancer cells

Yusha Li, Yuki Masuda, Yuzuha Miyazawa, DAISUKE TAKAHASHI, *Kazunobu Toshima

BIOORGANIC & MEDICINAL CHEMISTRY (Elsevier)  129   130371 - 130371 2025.08

Research paper (scientific journal), Joint Work, Accepted

Total Synthesis of Kanamycins

Kanae Hosomi, Banjo Imai, Naoto Takemura, Kazuki Senoo, Chigusa Hayashi, Masayuki Igarashi,*Kazunobu Toshima, *DAISUKE TAKAHASHI

CHEMISTRY-A EUROPEAN JOURNAL (Wiley-VCH)  31 ( 38 ) e202500685 (9 pages) 2025.04

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted

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Stereoselective Total Synthesis of α-Galacto-OligosaccharidesUsing Boron-Mediated Aglycon Delivery and Evaluation of their Immune-Enhancing Activities

Jikun Meng, Moeri Sagawa, *Kazunobu Toshima, *DAISUKE TAKAHASHI

CHEMBIOCHEM (Wiley-VCH)  26   e202401059 (6 pages) 2025.04

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted

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Photo-induced glycosylation using edible polyphenol ellagic acid

Hidenari Shigeta, Satomi Goi, DAISUKE TAKAHASHI, *Kazunobu Toshima

CARBOHYDRATE RESEARCH (Elsevier)  552   109461 (6 pages) 2025.03

Research paper (scientific journal), Joint Work, Accepted

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Creation of a New Macrolide Antibiotic against Non-tuberculous Mycobacterium Using Late-stage Boron-mediated Aglycon Delivery

Yuka Isozaki, Takumi Makikawa, Kosuke Kimura, Daiki Nishihara, Fujino, Yoshikazu Tanaka, Chigusa Hayashi, Yoshimasa Ishizaki, *Masayuki Igarashi, *Takeshi Yokoyama, *Kazunobu Toshima, *DAISUKE TAKAHASHI

SCIENCE ADVANCES (American Association for the Advancement of Science)  11 ( 10 ) eadt2352 (12 pages) 2025.03

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted

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A novel porphyrin-based theranostic agent activated by cysteine over-expressed in cancer cells shows promise for tumour-targeted monitoring and phototherapy

Fumihisa Ishida, Satoe Moriya, DAISUKE TAKAHASHI, *Kazunobu Toshima

BIOORGANIC & MEDICINAL CHEMISTRY (Elsevier)  121   118131 (9 pages) 2025.02

Research paper (scientific journal), Joint Work, Accepted

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Synthesis of Low-Molecular-Weight Fucoidan Analogue and Its Inhibitory Activities against Heparanase and SARS-CoV-2 Infection

Aoi Sugimoto, Tatsuki Koike, Yuya Kuboki, Sumika Komaba, Shuhei Kosono, Maniyamma Aswathy, Itsuki Anzai, Tokiko Watanabe, *Kazunobu Toshima, *DAISUKE TAKAHASHI

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (Wiley-VCH)  64 ( 6 ) e202411760 (7 pages) 2024.10

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted

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A novel photosensitizer based on hypocrellin B activated by cysteine over-expressed in cancer cells

Fumihisa Ishida, Rikuto Onishi, DAISUKE TAKAHASHI, *Kazunobu Toshima

ORGANIC & BIOMOLECULAR CHEMISTRY (Royal Society of Chemistry)  22   7187 - 7193 2024.08

Research paper (scientific journal), Joint Work, Accepted

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Designed Mannosylerythritol Lipid Analogues Exhibiting both Selective Cytotoxicity against Human Skin Cancer Cells and Recovery Effects on Damaged Skin Cells

Jikun Meng, Chihiro Yasui, Mai Shida, *Kazunobu Toshima, *DAISUKE TAKAHASHI

CHEMISTRY-A EUROPEAN JOURNAL (Wiley-VCH)  30   e202401319 (7 pages) 2024.05

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted

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Photo-Induced Glycosylation Using the Edible Polyphenol Curcumin

Satomi Goi, Hidenari Shigeta, DAISUKE TAKAHASHI, *Kazunobu Toshima

ORGANIC & BIOMOLECULAR CHEMISTRY (Royal Society of Chemistry)  22   5546 - 5551 2024.05

Research paper (scientific journal), Joint Work, Accepted

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Discovery of a Novel Photosensitizer Based on the Enediyne Antibiotic N1999A2 and Its Application as a Glutathione-Activatable Theranostic Agent

Kotono Matsunaga, Minami Takahashi, Tugumi Kagaya, DAISUKE TAKAHASHI, *Kazunobu Toshima

BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN (Chemical Society of Japan)  97 ( 5 ) uoae057 (9 pages) 2024.05

Research paper (scientific journal), Joint Work, Accepted

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Synthesis and Immunological Evaluation of Escherichia coli O1- Derived Oligosaccharide–Protein Conjugates toward Avian Pathogenic Escherichia coli O1 Vaccine Development

Katsunori Seki, Takumi Makikawa, *Kazunobu Toshima, *DAISUKE TAKAHASHI

SYNTHESIS (Georg Thieme Verlag KG)  56 ( 06 ) 953 - 965 2023.08

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted,  ISSN  0039-7881

Regioselective and Stereospecific β-Arabinofuranosylation by Boron-Mediated Aglycon Delivery

Kazuki Inaba, Yuna Naito, Mina Tachibana, *Kazunobu Toshima, *DAISUKE TAKAHASHI

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (Wiley-VCH)  62 ( 46 ) e202307015 (10 pages) 2023.07

Research paper (scientific journal), Joint Work, Last author, Corresponding author, Accepted,  ISSN  14337851

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Photoinduced Glycosylation Using a Diarylthiophene as an Organo Lewis Photoacid Catalyst

Naoki Otani, Kohei Higashiyama, Hayato Sakai, Taku Hasobe, *DAISUKE TAKAHASHI, *Kazunobu Toshima

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (Wiley-VCH)  26 ( 20 ) e202300287 (6 pages) 2023.04

Research paper (scientific journal), Joint Work, Corresponding author, Accepted,  ISSN  1434193X

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Destabilization of vitelline membrane outer layer protein 1 homolog (VMO1) by C‐mannosylation

Satoshi Yoshimoto, Takehiro Suzuki, Naoki Otani, DAISUKE TAKAHASHI, Kazunobu Toshima, Naoshi Dohmae, *Siro Simizu

FEBS OPEN BIO (Wiley-VCH)  13 ( 3 ) 490 - 499 2023.01

Research paper (scientific journal), Joint Work, Accepted,  ISSN  2211-5463

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Synthesis of Mannosylerythritol Lipid Analogues and their Self-Assembling Properties, Recovery Effects on Damaged Skin Cells, and Antibacterial Activity.

Takanori Kondo, Chihiro Yasui, Ikkei Miyajima, Taisuke Banno, Kouichi Asakura, Tokuma Fukuoka, Kazunori Ushimaru, Maito Koga, Azusa Saika, Tomotake Morita, Yoshiaki Takahashi, Chigusa Hayashi, Masayuki Igarashi, *DAISUKE TAKAHASHI, *Kazunobu Toshima

CHEMISTRY-A EUROPEAN JOURNAL (Wiley-VCH)  28 ( 55 ) e202201733 (7 pages) 2022.10

Research paper (scientific journal), Joint Work, Corresponding author, Accepted,  ISSN  09476539

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